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Collect. Czech. Chem. Commun. 1998, 63, 231-244
https://doi.org/10.1135/cccc19980231

Peptide Inhibitors of Aspartic Proteinases with Hydroxyethylene Isostere Replacement of Peptide Bond. I. Preparation of Four Diastereoisomeric (2R or 2S,4R or 4S,5S)-2-Benzyl-5-[(tert-butoxycarbonyl)amino]-4-hydroxy-6-phenylhexanoic Acids

Jaroslav Litera, Miloš Buděšínský, Ján Urban and Milan Souček

Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, 166 10 Prague 6, Czech Republic

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  • Ruan Shu-Tang, Luo Jie-Min, Du Yu, Huang Pei-Qiang: Asymmetric Vinylogous Mannich Reactions: A Versatile Approach to Functionalized Heterocycles. Org. Lett. 2011, 13, 4938. <https://doi.org/10.1021/ol2020384>
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  • Benedetti Fabio, Maman Paolo, Norbedo Stefano: New synthesis of 5-amino-4-hydroxy-2,6-dimethylheptanoic acid, a hydroxyethylene isostere of the Val-Ala dipeptide. Tetrahedron Letters 2000, 41, 10075. <https://doi.org/10.1016/S0040-4039(00)01773-1>
  • LITERA J., BUDESINSKY M., URBAN J., SOUCEK M.: ChemInform Abstract: Peptide Inhibitors of Aspartic Proteinases with Hydroxyethylene Isostere Replacement of Peptide Bond. Part 1. Preparation of Four Diastereoisomeric (2R or 2S,4R or 4S,5S)‐2‐Benzyl‐5‐ [(tert‐butoxycarbonyl)amino]‐4‐hydroxy‐6‐phenylhexanoic Acids. ChemInform 1998, 29. <https://doi.org/10.1002/chin.199828234>